Претрага
211 items
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Overcoming the Low Oral Bioavailability of Deuterated Pyrazoloquinolinone Ligand DK-I-60-3 by Nanonization: A Knowledge-Based Approach
Jelena R. Mitrović , Branka Divović-Matović, Daniel E. Knutson, Jelena B. Ðoković, Aleksandar Kremenović, Vladimir D. Dobričić, Danijela V. Randjelović, Ivana Pantelić, James M. Cook, Miroslav M. Savić, Snežana D. Savić (2021)Poor water solubility of new chemical entities is considered as one of the main obstacles in drug development, as it usually leads to low bioavailability after administration. To overcome these problems, the selection of the appropriate formulation technology needs to be based on the physicochemical properties of the drug and introduced in the early stages of drug research. One example of the new potential drug substance with poor solubility is DK-I-60-3, deuterated pyrazoloquinolinone, designed for the treatment of various neuropsychiatric ...Jelena R. Mitrović , Branka Divović-Matović, Daniel E. Knutson, Jelena B. Ðoković, Aleksandar Kremenović, Vladimir D. Dobričić, Danijela V. Randjelović, Ivana Pantelić, James M. Cook, Miroslav M. Savić, Snežana D. Savić. "Overcoming the Low Oral Bioavailability of Deuterated Pyrazoloquinolinone Ligand DK-I-60-3 by Nanonization: A Knowledge-Based Approach" in Pharmaceutics, MDPI, Basel, Switzerland (2021). https://doi.org/10.3390/pharmaceutics13081188 М21
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Organoselenium functionalized oxacycles as ligands in some trans-palladium(II) complexes: biological evaluation and interaction with small biomolecules
I. Raković, D. Ćoćić, O. Milošević-Djordjević, I. Radojević, M. N. Živanović, K. Virijević, J. Pavić, J. Tubić Vukajlović, A. Marković, J. S. Marjanović, M. D. Kostić, P. Čanović, A. Mijatović, V. M. Divac (2023)In this article, the biological evaluation and interaction of three selenium-based trans-palladium complexes (Pd–Se1, Pd–Se2, and Pd–Se3) with small biomolecules were performed. The UV–Vis kinetic studies on substitution reaction of synthesized complexes with selected biologically important N- and S-bonding ligands (LCys, GSH, L-Met, 50-GMP, L-His) has emphasized greater affinity of sulphur-based ligands for complex-binding, while the general order of the reactivity was L-Cys > GSH > L-Met > 50-GMP > L-His. The complex reactivity toward small biomolecules is influenced ...I. Raković, D. Ćoćić, O. Milošević-Djordjević, I. Radojević, M. N. Živanović, K. Virijević, J. Pavić, J. Tubić Vukajlović, A. Marković, J. S. Marjanović, M. D. Kostić, P. Čanović, A. Mijatović, V. M. Divac. "Organoselenium functionalized oxacycles as ligands in some trans-palladium(II) complexes: biological evaluation and interaction with small biomolecules" in Journal of Coordination Chemistry, Informa UK Limited (2023). https://doi.org/10.1080/00958972.2023.2256934 М23
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Optimizacija reznih elemenata rotornog bagera pri otkopavanju uglja
Jovančić Predrag, Ignjatović Dragan, Novaković Dragan. "Optimizacija reznih elemenata rotornog bagera pri otkopavanju uglja" in V Međunarodna konferencija UGALJ 1, Zlatibor:Rudarsko-geološki fakultet (2011): 124-138 M33
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Selective separation processes of complex auriferous minerals
Tomanec Rudolf, Lazić Predrag (2010)Tomanec Rudolf, Lazić Predrag. "Selective separation processes of complex auriferous minerals" in Proceedings of Workshop – Vyskum v oblasti otpadu jako nahrady primarnich surovinovych zdroju, Ostrava:VŠB-Technical University of Ostrava (2010): 135-142 M33
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Uticaj promena klime na procenu hazarda od klizišta na putnoj mreži Srbije
Abolmasov Biljana (2017)Abolmasov Biljana. "Uticaj promena klime na procenu hazarda od klizišta na putnoj mreži Srbije" in Zbornik radova V naučno stručnog savetovanja Put I životna sredina, Vršac 28-29 septembar 2017 1, Beograd:VIA VITA (2017): 18-31 M61
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Примена методе раздвојених елемената у подземној експлоатацији
Lapčević Veljko, Torbica Slavko (2017)Lapčević Veljko, Torbica Slavko. "Примена методе раздвојених елемената у подземној експлоатацији" in Зборник радова са V научно - стручног скупа „Подземна експлоатација минералних сировина 2017“, Univerzitet u Beogradu - Rudarsko-geološki fakultet (2017): 37-42 M63
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Hidrogeološka prospekcija u jugoistočnoj Mongoliji
Ristić-Vakanjac Vesna, Vakanjac Boris, Kondžulović Rajko. "Hidrogeološka prospekcija u jugoistočnoj Mongoliji" in Zapisnici Srpskog geološkog društva, Beograd, Srbija:Srpsko geološko društvo (2014): 159-172 M53
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On Linear Combinations of the Chebyshev Polynomials
Stankov Dragan (2015)Stankov Dragan. "On Linear Combinations of the Chebyshev Polynomials" in Publications de lInstitut Mathématique 111 no. 97, Beograd:Matematički institut SANU (2015): 57-67. https://doi.org/DOI: 10.2298/PIM150220001S M23
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Nova saznanja o geologiji Vrdničkog ugljenog basena (severna Srbija)
Rundić Ljupko, Knežević Slobodan, Rakijaš Milovan, Kukavica Marija. "Nova saznanja o geologiji Vrdničkog ugljenog basena (severna Srbija)" in Zbornik radova V Savjetovanja geologa BiH *CD-ROM, Sarajevo, BiH:Udruženje geologa BiH (2013): 330-348 M33
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Reclamation methods and their outcomes in Serbian mining basins
Ranđelović Dragana (2017)Ranđelović Dragana. "Reclamation methods and their outcomes in Serbian mining basins" in Book of Abstracts of 2nd International and 14th National Congress of Soil Science Society of Serbia Solutions and Projections for Sustainable Soil Management, :Soil Science Society of Serbia (2017): 56-57 M32
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Middle Jurassic terebratulide brachiopods from the Jordan Valley (northwestern Jordan)
U radu je izvršena revizija i detaljan opis srednjojurskih brahiopoda Jordanske doline, a takodje su izdvojeni i novi taksoni. Sa profila Arda iz gornjeg bata (Hamam formacija) i donjeg keloveja (Muganija formacija) odredjeni su novi rod i vrsta Jordanithyris ardainensis. Iz gornjeg bata Hamam formacije (krečnjaci, dolomiti, peščari i laporci) izdvojena je vrsta Ptyctothyris quillyensis. Zajednica koju čine Arabatia bihinensis, Ectyphoria sinaiensis, Ptyctothyris quillyensis, Dorsoplicathyris dorsoplicata i Tubithyris jurayfahiensis potiče iz donjokelovejskih krečnjaka sa proslojcima laporaca Muganija formacije. Brahiopodi ...Howard R. Feldman, Barbara V. Radulović, Vladan J. Radulović, Fayez Ahmadc. "Middle Jurassic terebratulide brachiopods from the Jordan Valley (northwestern Jordan)" in Historical Biology, Taylor & Francis (2021). https://doi.org/10.1080/08912963.2019.1625347 М21
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Crystallographic, spectroscopic, thermal and computational studies of polymeric cobalt(II)–mellitate complex with 2,2′-bipyridine
Orange single crystals of new polymeric cobalt(II) complex {[Co(bipy)(H2O)4]2[Co(μ-mell)(H2O)2]·10H2O}n, 1, were synthesized by slow evaporation method at room temperature (bipy = 2,2′-bipyridine, mell = hexaanion of mellitic acid) and its crystal structure was determined by single-crystal X-ray diffraction. The complex 1 was characterized based on elemental analysis, FTIR spectroscopy and thermal (TG/DTA) analysis followed by computational analysis of noncovalent interactions and quantum chemical calculations of interaction energies. In 1, two crystallographically different Co(II) atoms adopt a deformed octahedral geometry, ...Lidija Radovanović, Dušan P. Malenov, Marko V. Rodić, Aleksandar Kremenović, Jelena Rogan. "Crystallographic, spectroscopic, thermal and computational studies of polymeric cobalt(II)–mellitate complex with 2,2′-bipyridine" in Journal of Molecular Structure, Elsevier BV (2021). https://doi.org/10.1016/j.molstruc.2021.132202 М22
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Primena savremenih geodetskih tehnologija u funkciji određivanja zapremina na površinskim kopovima uglja
Pandžić Slobodan, Milutinović Aleksandar, Ganić Aleksandar, Pandžić Jelena. "Primena savremenih geodetskih tehnologija u funkciji određivanja zapremina na površinskim kopovima uglja" in V Međunarodna konferencija UGALJ 2011 1, Zlatibor:Rudarsko-geološki fakultet, Beograd (2011): 244-253 M63
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Hydrodynamic calculation of the screen section 1 at the opencast coal mine Drmno
Šubaranović Tomislav, Pavlović Vladimir, Polomčić Dušan. "Hydrodynamic calculation of the screen section 1 at the opencast coal mine Drmno" in V International Conference COAL, Zlatibor: (2011): 355-361 M33
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BPUBS: Informacioni sistem za istražne radove ugljenih basena Srbije
Gojak Zorica, Mitrović Slobodan, Stanković Ranka, Kitanović Olivera. "BPUBS: Informacioni sistem za istražne radove ugljenih basena Srbije" in Zbornik radova V međunarodne konferencije UGALJ 2011, :Jugoslovenski komitete za površinsku eksploataciju (2011): 66-73 M63
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3D Hydrodinamic model of open pit mine “Polje E” (Kolubara coal basin)
Polomčić Dušan, Bajić Dragoljub (2011)Polomčić Dušan, Bajić Dragoljub. "3D Hydrodinamic model of open pit mine “Polje E” (Kolubara coal basin)" in Proceedings of the V International Conference “Coal 2011”, Zlatibor, Serbia, 19-22 October, 2011, Belgrade:Yugoslav Opencast Mining Committee (2011): 320-330 M33
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Procena rizika od klizišta na putnoj mreži opštine Krupanj
Marjanović Miloš, Abolmasov Biljana, Milenković Svetozar. "Procena rizika od klizišta na putnoj mreži opštine Krupanj" in Zbornik radova V naučno stručnog savetovanja Put I životna sredina, Vršac 28-29 septembar 2017 1, Beograd:VIA VITA (2017): 491-500 M63
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DIMENZIONISANjE POPREČNOG PRESEKA I IZBOR OBLOGE HIDROTEHNIČKOG TUNELA “VLADIKINE PLOČE”
Crnogorac Luka, Tokalić Rade (2017)Crnogorac Luka, Tokalić Rade. "DIMENZIONISANjE POPREČNOG PRESEKA I IZBOR OBLOGE HIDROTEHNIČKOG TUNELA “VLADIKINE PLOČE”" in Zbornik radova sa V naučno - stručnog skupa „Podzemna eksploatacija mineralnih sirovina 2017“, :Univerzitet u Beogradu – Rudarsko – geološki fakultet (2017): 28-36 M61
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Uticaj padavina na hidrohemijski režim vrela Banje kod Petnice
Golubović Radisav, Ristić-Vakanjac Vesna, Papić Petar. "Uticaj padavina na hidrohemijski režim vrela Banje kod Petnice" in Zapisnici Srpskog geološkog društva, Beograd, Srbija:Srpsko geološko društvo (2014): 145-158 M53
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Influence of Galena Grain Size and Collector Concentration on Recovery and Flotation Rate
Cvetićanin Lidija, Lazić Predrag, Vučinić Dušica. "Influence of Galena Grain Size and Collector Concentration on Recovery and Flotation Rate" in Journal of Mining Science 54 no. 3, Switzerland:Springer Nature Switzerland AG (2018): u stampi-u stampi M23